TaiClone24 [TaiClone] Elagolix sodium [TaiClone] Elagolix sodium tcsc0003317 Specifications Purity / Grade >98% Solubility 10 mM in DMSO Smiles smiles Misc Information Alternative Names NBI-56418 sodium Observed Molecular Weight 653.57 Product Description Elagolix sodium is a human GnRH receptor (GnRHR) antagonist with an IC50 and Ki of 0.25 and 3.7 nM, respectively. IC50 & Target: IC50: 0.25 nM (GnRHR)[1] Ki: 3.7 nM (GnRHR)[2] In V.. 2020. 10. 19. [TaiClone] NS 1738 [TaiClone] NS 1738 tcsc0003117 Product Description NS1738 is a novel positive allosteric modulator of the α7 nAChR, with respect to positive modulation of α7 nAChR (EC50=3.4 μM in oocyte experiments). IC50 & Target: EC50: 3.4 μM (α7 nAChR, in oocyte experiments)[1] In Vitro: NS1738 acts by increasing the peak amplitude of acetylcholine (ACh)-evoked currents at all concentrations; thus, it increa.. 2020. 8. 25. [TaiClone] GSK-269984A [TaiClone] GSK-269984A tcsc0003376 Specifications Purity / Grade >98% Solubility 10 mM in DMSO Smiles smiles Misc Information Observed Molecular Weight 429.22 Product Description GSK-269984A is a Prostaglandin E2 Receptor 1 (EP1) antagonist with a pIC50 of 7.9. IC50 & Target: pIC50: 7.9 (Prostaglandin E2 Receptor 1 (EP1))[1] In Vitro: Results from [3H]-PGE2 binding assay in CHO cells overexpress.. 2020. 8. 5. [Taiclone] Active Vascular Endothelial Growth Factor A (VEGFA) [Taiclone] Active Vascular Endothelial Growth Factor A (VEGFA) tcup82 Product Description Eukaryotic expression Information Application Cell culture Activity Assays. Species Rattus norvegicus (Rat) Specifications Source 293F cell Purity / Grade > 97% Amino Acids Ala27~Arg190 Misc Information SwissProt P16612 Predicted Molecular Weight 20.8kDa Observed Molecular Weight 22kDa Tags N-terminal His Tag 2020. 7. 15. [TaiClone] Emicerfont [TaiClone] Emicerfont tcsc0003315 Specifications Purity / Grade>98% Solubility10 mM in DMSO Smilessmiles Misc Information Alternative NamesGW876008 Observed Molecular W Product Description Emicerfont is a corticotropin-releasing factor type 1 (CRF1) receptor antagonist with an IC50 of 66 nM. IC50 & Target: IC50: 66 nM (CRF1 receptor)[1] In Vitro: Emicerfont is a corticotropin-releasing factor ty.. 2020. 6. 1. [TaiClone] Vofopitant [TaiClone] Vofopitant tcsc0003109 Specifications Purity / Grade >98% Solubility 10 mM in DMSO Smiles smiles Misc Information Alternative Names GR 205171 Observed Molecular Weight 432.44 2020. 4. 29. [TaiClone] Temanogrel [TaiClone] Temanogrel tcsc0002653 Specifications Purity / Grade >98% Solubility DMSO : 125 mg/mL (286.37 mM; Need ultrasonic) Smiles smiles Misc Information Alternative Names APD791 Observed Molecular Weight 436.5 Information CAS No 887936-68-7 Formula C24H28N4O4 Clinical Information clinicalinformation Pathway Neuronal Signaling GPCR/G Protein Target 5-HT Receptor 5-HT Receptor 2020. 4. 13. [TaiClone] NS 1738 [TaiClone] NS 1738 CAS No 501684-93-1 Formula C14H9Cl2F3N2O2 Clinical Information Pathway Neuronal Signaling Membrane Transporter/Ion Channel Targetn AChR nAChR Purity / Grade >98% Solubility DMSO : ≥ 300 mg/mL (821.63 mM) Smiles smiles Misc Information Alternative Names NSC 213859 Observed Molecular Weight 365.13 Product Description NS1738 is a novel positive allosteric modulator of the α7 nACh.. 2020. 3. 30. 이전 1 2 3 다음
